著者
Jiao Jiao Kei Murakami Kenichiro Itami
出版者
(社)日本化学会
雑誌
Chemistry Letters (ISSN:03667022)
巻号頁・発行日
pp.160133, (Released:2016-02-25)
被引用文献数
14

Methods that can directly arylate pyridines have significant potential in synthetic chemistry. Herein, we present a palladium-catalyzed C–H arylation of pyridines with aryl triflates that occurs regioselectively at the C3 positions of pyridine core. A variety of aryl triflates and pyridines were applicable to the reaction to provide C3-arylated pyridines regardless of sterics or electronics of the pyridine cores.